Drug |
Therapeutic area |
Gene |
Relevance class |
pimozid |
psychiatry |
CYP2D6 |
required |
tetrabenazin |
neurology |
CYP2D6 |
required |
siponimod |
neurology |
CYP2C9 |
required |
atazanavir |
infectiology |
UGT1A1, (CYP2C19) |
recommended |
azathioprin |
rheumatology |
TPMT1, NUDT15 |
recommended |
mercaptopurin |
oncology |
TPMT1, NUDT15 |
recommended |
amitriptylin |
psychiatry |
CYP2D6, CYP2C19 |
actionable |
aripiprazol |
psychiatry |
CYP2D6 |
actionable |
atomoxetin |
psychiatry |
CYP2D6 |
actionable |
atorvastatin |
cardiology |
SLCO1B1 |
actionable |
brexpiprazol |
psychiatry |
CYP2D6 |
actionable |
capecitabin |
oncology |
DPYD |
actionable |
carisoprodol |
rheumatology |
CYP2C19 |
actionable |
carvedilol |
cardiology |
CYP2D6 |
actionable |
celecoxib |
rheumatology |
CYP2C9 |
actionable |
cevimelin |
autoimmune disease |
CYP2D6 |
actionable |
citalopram |
psychiatry |
CYP2C19, (CYP2D6) |
actionable |
clobazam |
neurology |
CYP2C19 |
actionable |
clomipramin |
psychiatry |
CYP2D6, CYP2C19 |
actionable |
clopidogrel |
cardiology |
CYP2C19 |
actionable |
clozapin |
psychiatry |
CYP2D6 |
actionable |
codein |
pain therapy |
CYP2D6, OPRM1, CYP3A4 |
actionable |
darifenacin |
urology |
CYP2D6 |
actionable |
desipramin |
psychiatry |
CYP2D6, CYP2C19 |
actionable |
doxepin |
psychiatry |
CYP2D6, (CYP2C19) |
actionable |
efavirenz |
infectiology |
CYP2B6 |
actionable |
fesoterodin |
urology |
CYP2D6 |
actionable |
fluorouracil |
oncology |
DPYD |
actionable |
iloperidon |
psychiatry |
CYP2D6 |
actionable |
imipramin |
psychiatry |
CYP2C6, CYP2C19 |
actionable |
nortriptylin |
psychiatry |
CYP2D6, CYP2C19 |
actionable |
pantoprazol |
gastroenterology |
CYP2C19 |
actionable |
perphenazin |
psychiatry |
CYP2D6 |
actionable |
phenytoin |
neurology |
CYP2C9 |
actionable |
propafenon |
cardiology |
CYP2D6 |
actionable |
simvastatin |
cardiology |
SLCO1B1 |
actionable |
tamoxifen |
oncology |
CYP2D6, CYP3A4 |
actionable |
thioridazin |
psychiatry |
CYP2D6 |
actionable |
tioguanin |
oncology |
TPMT1, NUDT15 |
actionable |
tramadol |
pain therapy |
CYP2D6 |
actionable |
trimipramin |
psychiatry |
CYP2D6, CYP2C19 |
actionable |
voriconazol |
infectiology |
CYP2C19 |
actionable |
vortioxetin |
psychiatry |
CYP2D6 |
actionable |
warfarin |
cardiology |
CYP2C9, VKORC1, CYP4F2 |
actionable |
acenoumarol |
cardiology |
CYP2C9, VKORC1,CYP4F2 |
informative |
diclofenac |
rheumatology |
CYP2C9 |
informative |
escitalopram |
psychiatry |
CYP2C19 |
informative |
flecainid |
cardiology |
CYP2D6 |
informative |
fluribiprofen |
rheumatology |
CYP2C9 |
informative |
fluvoxamin |
psychiatry |
CYP2D6 |
informative |
haloperidol |
psychiatry |
CYP2D6 |
informative |
ibuprofen |
rheumatology |
CYP2C9 |
informative |
lansoprazol |
gastroenterology |
CYP2C19 |
informative |
methoxyfluran |
anaesthesiology |
CACNA1S, RYR1 |
informative |
metoprolol |
cardiology |
CYP2D6 |
informative |
mirtazapin |
psychiatry |
CYP2D6 (CYP1A2, CYP3A4) |
informative |
morphin |
pain therapy |
OPRM1 |
informative |
olanzapin |
psychiatry |
CYP1A2, (CYP2D6) |
informative |
omeprazol |
gastroenterology |
CYP2C19 |
informative |
ondansetron |
oncology |
CYP2D6 |
informative |
oxycodon |
pain therapy |
CYP2D6 (CYP2C19) |
informative |
paroxetin |
psychiatry |
CYP2D6 |
informative |
phenprocoumon |
cardiology |
CYP2C9, VKORC1,CYP4F2 |
informative |
piroxicam |
rheumatology |
CYP2C9 |
informative |
propofol |
anaesthesiology |
CYP2B6 |
informative |
risperidon |
psychiatry |
CYP2D6 |
informative |
rosuvastatin |
cardiology |
SLCO1B1 |
informative |
sertralin |
psychiatry |
CYP2C19 |
informative |
tacrolismus |
transplantation |
CYP3A5, POR (CYP3A4) |
informative |
tropisetron |
oncology |
CYP2D6 |
informative |
venlafaxin |
psychiatry |
CYP2D6 |
informative |
zuclopenthixol |
psychiatry |
CYP2D6 |
informative |