Ligand
ΔΔLog(Emax/EC50)
Pathway 1 Emax (%) Pathway 2 Emax (%) Pathway 1 pEC50 Pathway 2 pEC50 Pathway 1 CRC slope Pathway 2 CRC slope
Ligand A
- (reference ligand, unbiased by definition)
100
100
8.3
9.0
0.9
1.1
Ligand B 0.8 83 97 8.7 10.1 1.0 1.2